Platform Evidence

Platform Evidence & Applications

Molecule studies completed to date provide evidence of the breadth and applicability of the Mirai™ architecture. They should not be interpreted as independently developed product assets unless specifically stated.

How to read the evidence

Independently tested in-vitro proof of conceptTeam formulation expertisePotential future application

Pre-Clinical Development

Budesonide and fluticasone propionate formulations have generated RLD-comparable in-vitro aerosol-performance signals through the Mirai™ development chassis during independent Intertek testing. Ciclesonide, a repurposed candidate for eosinophilic esophagitis (EoE), has separately completed independent proof-of-concept testing at Intertek (emitted dose and APSD by extended cascade impaction, across two batches). Formulation details and reports are available on request and on signing of a CDA.

API (INN)Therapeutic AreaAnalyticalStatus
BudesonideICS - Inhaled CorticosteroidIndependently testedAsthmaDDU, APSD (NGI)POC - Overlaid RLD
Fluticasone propionateICS - Inhaled CorticosteroidIndependently testedAsthmaDDU, APSD (NGI)POC - Matched RLD
CiclesonideICS - Inhaled CorticosteroidIndependently testedEoEDDU, APSD (CI)POC - Repurposed drug

POC = Proof of Concept · DDU = Dose Delivered Uniformity · APSD = Aerodynamic Particle Size Distribution (incl. MMAD, Mass Median Aerodynamic Diameter) · NGI = Next Generation Impactor · CI = Cascade Impactor · EoE = Eosinophilic Esophagitis · RLD = Reference Listed Drug

Reflects in-vitro device performance (pre-clinical); no human trials have been conducted.

See the full budesonide performance data (APSD vs. RLD) →

Formulation Capability

Team formulation expertise

Given the encouraging pre-clinical results - completely matching the APSD of the RLD for budesonide and performing very closely with fluticasone propionate at first attempt - Knightpoint has the expertise to develop a broad range of dry-powder formulations across the major respiratory classes - for example tiotropium bromide (COPD), albuterol (rescue), or zanamivir (antiviral).

Partnership Opportunity: Generic Triple-Combination Therapy

Potential future application

Knightpoint is open to a partnership opportunity for any client seeking to develop the next generation of triple-therapy medicines currently on the market. Through in-house, in-depth technical expertise across the API / formulation / device eco-system, Knightpoint can develop - for example - umeclidinium / vilanterol / fluticasone furoate in a single-capsule system delivered through the Mirai™ platform.

Formulation Breadth

Representative Molecules and Platform Applications

The molecules below illustrate the breadth of formulation capability across every major respiratory class, from inhaled corticosteroids to antimicrobials. They are representative examples of what the Mirai™ platform can formulate - not a portfolio of active pharmaceutical ingredients owned or licensed by Knightpoint.

Inhaled Corticosteroids (ICS)

Anti-inflammatory agents for respiratory conditions

Fluticasone Furoate
Fluticasone Propionate
Budesonide
Ciclesonide
Mometasone Furoate
Beclomethasone Dipropionate

Long-Acting Muscarinic Antagonists (LAMA)

Bronchodilators for COPD and respiratory conditions

Umeclidinium
Tiotropium Bromide
Glycopyrronium Bromide

Long-Acting Beta-Agonists (LABA)

Bronchodilators for asthma and COPD

Vilanterol
Formoterol Fumarate Dihydrate
Salmeterol Xinafoate
Indacaterol Maleate
Salbutamol Sulphate

Antimicrobials

Inhaled antibiotics for respiratory infections

Tobramycin

Formulation–Device Integration Capability

Knightpoint develops the formulation and the device together as one system. This integrated capability - not formulation offered in isolation - is what lets each combination product be optimised end-to-end on the Mirai™ platform.

DPI Formulations

Dry powder inhaler formulation development optimized for the Mirai™ platform.

Combination Products

Multi-component formulations including dual and triple-combination therapies.

Stability & Characterisation

Formulation stability and in-vitro aerosol characterisation, evaluated on the Mirai™ device.

FDA Combination Product Pathway

Products built on the Mirai™ device follow the FDA combination product regulatory pathway - integrated drug + device products evaluated as a single system. This approach enables:

  • Optimized device-formulation integration
  • Unified regulatory submission
  • Clear primary mode of action designation
  • Potential for expedited development timelines

Our Expertise

Corticosteroids
ICS formulation development
LAMAs
Long-acting muscarinic antagonists
LABAs
Long-acting beta-agonists
Triple Combinations
ICS/LAMA/LABA expertise

Strategic Opportunities

The Mirai™ patent estate, device architecture, development evidence and associated know-how are available for confidential strategic discussion. Selected licensing and programme structures may also be considered.